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Publications
Publications
  • Wojciechowski P, Szereda-Przestaszewska M, Lipkowski AW. (2007) Supranodose vagotomy eliminates respiratory depression evoked by dermorphin in anaesthetized rats. Eur J Pharmacol. 563:209-212
  • Ioja E, Tourwé D, Kertész I, Tóth G, Borsodi A, Benyhe S. (2007) Novel diastereomeric opioid tetrapeptides exhibit differing pharmacological activity profiles. Brain Res Bull. 74:119-129
  • Łazarczyk M, Matyja E. Lipkowski A. (2007) Substance P and its receptors -- a potential target for novel medicinesin malignant brain tumour therapies (mini-review). Folia Neuropathol.45:99-107.
  • Pasquinucci L, Iadanza M, Marrazzo A, Prezzavento O, Ronsisvalle S, Scoto GM, Parenti C, De Luca L, Ronsisvalle G. (2007) New benzomorphan derivatives of MPCB as MOP and KOP receptor ligands.  Pharmazie, 62: 813-824
  • Niedzialek D, Urbanczyk-Lipkowska Z. (2007) New Crystalline form of 7-amino-4-methylcoumarin (coumarin 120) – a polymorph with (1:1) valence tautomers” CrystEngComm, 9: 735-739
  • Ballet S, Misicka A, Kosson P, Lemieux C, Chung NN, Schiller PW, Lipkowski AW, Tourwé D (2008) Blood-Brain Barrier Penetration by Two Dermorphin Tetrapeptide Analogues: Role of Lipophilicity vs Structural Flexibility. J Med Chem. 51: 2571-2574
  • Pulka K, Kulis P, Tymecka D, Frankiewicz L, Wilczek, Kozminski W, Misicka A (2008) Diastereoselective Pictet-Spengler condensation of tryptophan with a-amino aldehydes as chiral carbonyl components, Tetrahedron 64: 1506-1514
  • Tömböly Cs, Ballett S, Feytens D, Kövér KE, Borics A, Lovas S, Al-Khrasani M, Fürst Z, Tóth G, Benyhe S, Tourwé D. (2008) Endomorphin-2 with a β-Turn Backbone Constraint Retains the Potent μ Opioid Receptor Agonist Properties J.Med.Chem. 51., 173-177.
  • Szemenyei E, Barna I, Mergl Z, Keresztes A, Darula Z, Kató E, Tóth G, Rónai A. (2008) Detection of a novel immonoreactive endomorphin 2-like peptide in rat brain extracts 22 Reg. Peptides 148: 54-61
  • Keresztes A, Szűcs M, Borics A, Kövér KE, Forró E, Fülöp F, Tömböly C,Péter A, Páhi A, Fábián G, Murányi M, Tóth G. (2008) New Endomorphin Analogues Containing Alicyclic β-Amino Acids: Influence on Bioactive Conformation and Pharmacological Profile J. Med. Chem. 51: 4270-4279
  • Botros M, Johanson T, Zhau Q, Lindeberg G, Tömböly C, Tóth G, Le Greves P, Nyberg F,  Hallberg M. (2008) Endomorphins interact with the substance P (SP) aminoterminal SP 1-7 binding in the ventral tegmental area of the brain Pepides 29: 1820-1824
  • Gramowski A, Schröder O, Jügelt K, Lipkowski A, Misicka-Kesik A, Weiss DG. (2008) Drug development of new synthetic peptides for cancer pain treatment: Electrophysiological profiling of the opioid receptor system. 6th Int. Meeting on Substrate-Integrated Microelectrodes, 2008: 217-220
  • Rónai A, Király K, Szebeni A, Szemenyei E, Prohászka Z, Darula Z, Tóth G, Till I, Szalai B,  Kató E, Barna I. (2009) Immunoreactive endomorphin-2 is genarated extracellularly in rat isolated L4,5 dorsal root ganglia by DPP-IV Reg Peptides 157: 1-2
  • De Wachter R, Brans L, Ballet S, Van den Eynde I, Feytens D, Keresztes A, Tóth G, Urbanczyk-Lipkowska Z, Tourwé D. (2009) Influence of ring substitution on the conformation and b-turn mimicry of 4-amino-1,2,4,5-tetrahydro-2 -benzazepin-3-one peptide mimetics Tetrahedron 65: 2266-2278
  • Borics A, Tóth G. (2009) Structural comparison of b-opioid receptor selective peptides confirmed four parameters of bioactivity. J. Mol. Graph. Model., in press.
  • Leontiadis LJ, Papakonstantinou M, Georgoussi Z. (2009). Regulator of G protein signaling 4 confers selectivity to specific G proteins to modulate μ- and δ-opioid receptor signaling.  Cell Sign 21: 1218-1228.
  • Lukowiak M, Kosson P,  Hennink WE, Lipkowski AW. (2009) The synthesis and pharmacological properties of new fluorescent opioid peptide analogue.Pharmacol Rep. 61: 517-521
  • Wojciechowski P, Szereda-Przestaszewska M, Lipkowski AW. (2009) Respiratory and cardiovascular effects of biphalin in anesthetized rats., Eur J Pharmacol. 602: 50-53
  • Berkecz R, Ilisz I, Misicka A, Tymecka D, Fülöp F, Choi HJ, Hyun MH, Péter A. (2009) HPLC enantioseparation of ß2-homoamino acids using crown ether-based chiral stationary phase. J Sep Sci 3: 981-987
  • Pataj Z, Berkecz R, Ilisz I, Misicka A, Tymecka D, Fulop F, Armstrong D, Peter A. (2009) High-Performance Liquid Chromatographic Chiral Separation of b2-Homo-Amino Acids, Chirality 21: 787-798
  • Ballet S,  Feytens D, De Wachter R, De Vlaeminck M, Marczak EW, Salvadori S,  de Graaf C,  Rognan D, Negri L, Lattanzi R, Lazarus LH, Tourwé D, Balboni G. (2009) Conformationally constrained opioid ligands: the Dmt-Aba and Dmt-Aia versus Dmt-Tic scaffold.Bioorg & Med Chem Lett. 19: 433-437.
  • Polcyn P, Janiszewska J, Lipkowski, AW,  Urbanczyk-Lipkowska Z. (2009) Syntheses, methods of identification and selected medical applications of dendrimers. Polimery, 54: 407-41
  • De Wachter R, Brans L, Ballet S, Van den Eynde I, Feytens D, Keresztes A, Toth G, Urbanczyk-Lipkowska Z, Tourwe D (2009) Influence of ring substitution on the conformation and beta-turn mimicry of 4-amino-1,2,4,5-tetrahydro-2-benzazepin-3-one peptide mimetics.Tetrahedron 65: 2266-2278
  • Polcyn P, Jurczak M, Rajnisz A, Solecka J, Urbanczyk-Lipkowska Z. (2009) Design of antimicrobially active small amphiphilic peptide dendrimers Molecules 14: 3881-3905
 


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  • Two awards in Brussels
  • Diploma for Young Investigator at Greifswald

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